Jérôme E.G. Guillemont: search on Z-Library

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1

Diarylquinolines target subunit c of mycobacterial ATP synthase

Koul, Anil, Dendouga, Najoua, Vergauwen, Karen, Molenberghs, Brenda, Vranckx, Luc, Willebrords, Rudy, Ristic, Zorica, Lill, Holger, Dorange, Ismet, Guillemont, Jerome

Journal:

Nature Chemical Biology

Year:

2007

Language:

english

File:

PDF, 434 KB

english, 2007

2

4-Benzyl and 4-Benzoyl-3-dimethylaminopyridin-2(1H)-ones: In Vitro Evaluation of New C-3-Amino-Substituted and C-5,6-Alkyl-Substituted Analogues against Clinically Important HIV Mutant Strains

Benjahad, Abdellah, Croisy, Martine, Monneret, Claude, Bisagni, Emile, Mabire, Dominique, Coupa, Sophie, Poncelet, Alain, Csoka, Imre, Guillemont, Jérôme, Meyer, Christophe

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 457 KB

english, 2005

3

Novel Procedure for the Coupling of Sterically Hindered Electron-Deficient Anilines to the 6-Position of the Purine Core

Leenders, Ruben, Heeres, Jan, Vandenput, Dirk, Guillemont, Jérôme, Lewi, Paul

Journal:

Synthetic Communications

Year:

2011

Language:

english

File:

PDF, 265 KB

english, 2011

4

4-Benzyl- and 4-Benzoyl-3-dimethylaminopyridin-2(1 H )-ones, a New Family of Potent Anti-HIV Agents: Optimization and in Vitro Evaluation against Clinically Important HIV Mutant Strains

Benjahad, Abdellah, Courté, Karine, Guillemont, Jérôme, Mabire, Dominique, Coupa, Sophie, Poncelet, Alain, Csoka, Imre, Andries, Koen, Pauwels, Rudi, de Béthune, Marie-Pierre, Monneret, Claude, Bisagn

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 264 KB

english, 2004

5

A new prenylation method using the lithium enolate of prenal. Reaction with aldehydes and α,β-unsaturated aldehydes.

Lucette Duhamel, Jerôme Guillemont, Jean-Marie Poirier, Pierre Chabardes

Journal:

Tetrahedron Letters

Year:

1991

Language:

english

File:

PDF, 161 KB

english, 1991

6

A new prenylation method using the lithium enolate of prenal. Reaction with polyunsaturated aldehydes. A short access to retinal.

Lucette Duhamel, Jerôme Guillemont, Jean-Marie Poirier, Pierre Chabardes

Journal:

Tetrahedron Letters

Year:

1991

Language:

english

File:

PDF, 84 KB

english, 1991

7

ChemInform Abstract: A Novel Route to 2,4-Dianilino-Substituted Pyrimidines.

Ruben Leenders, Jan Heeres, Jerome Guillemont, Paul Lewi

Journal:

Year:

2010

File:

PDF, 46 KB

2010

8

A novel route to 2,4-dianilino-substituted pyrimidines

Ruben Leenders, Jan Heeres, Jérôme Guillemont, Paul Lewi

Journal:

Tetrahedron Letters

Year:

2010

Language:

english

File:

PDF, 255 KB

english, 2010

9

Synthesis of Novel Diarylpyrimidine Analogues and Their Antiviral Activity against Human Immunodeficiency Virus Type 1

Guillemont, Jerome, Pasquier, Elisabeth, Palandjian, Patrice, Vernier, Daniel, Gaurrand, Sandrine, Lewi, Paul J., Heeres, Jan, de Jonge, Marc R., Koymans, Lucien M. H., Daeyaert, Frits F. D., Vinkers,

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 174 KB

english, 2005

10

Diarylquinolines, synthesis pathways and quantitative structure–activity relationship studies leading to the discovery of TMC207

Guillemont, Jerome, Meyer, Christophe, Poncelet, Alain, Bourdrez, Xavier, Andries, Koen

Journal:

Future Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 1.97 MB

english, 2011

11

Structure–activity relationship in the 3-iodo-4-phenoxypyridinone (IOPY) series: The nature of the C-3 substituent on anti-HIV activity

Abdellah Benjahad, Said Oumouch, Jerôme Guillemont, Elisabeth Pasquier, Dominique Mabire, Koen Andries, Chi Hung Nguyen, David S. Grierson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 188 KB

english, 2007

12

Bromation des enamines du prénal et du crotonaldéhyde. Voie d'accès aux ω-bromo aldéhydes et ω-bromo acétals correspondants.

Lucette Duhamel, Jerôme Guillemont, Jean-Marie Poirier, Pierre Chabardes

Journal:

Tetrahedron Letters

Year:

1992

File:

PDF, 256 KB

1992

13

Selection of a Respiratory Syncytial Virus Fusion Inhibitor Clinical Candidate, Part 1: Improving the Pharmacokinetic Profile Using the Structure−Property Relationship

Bonfanti, Jean-François, Doublet, Frédéric, Fortin, Jérôme, Lacrampe, Jean, Guillemont, Jérôme, Muller, Philippe, Queguiner, Laurence, Arnoult, Eric, Gevers, Tom, Janssens, Peggy, Szel, Heidi, Willebr

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 256 KB

english, 2007

14

Reduction of Alkynyl α-Hydroxy Esters: Stereoselective α-Ketol Rearrangement

Thomas Hameury, Véronique Bellosta, Jérôme Guillemont, Luc Van Hijfte, Janine Cossy

Journal:

European Journal of Organic Chemistry

Year:

2010

Language:

english

File:

PDF, 437 KB

english, 2010

15

Essentiality of FASII pathway for Staphylococcus aureus

Balemans, Wendy, Lounis, Nacer, Gilissen, Ron, Guillemont, Jerome, Simmen, Kenny, Andries, Koen, Koul, Anil

Journal:

Year:

2010

Language:

english

File:

PDF, 240 KB

english, 2010

16

The challenge of new drug discovery for tuberculosis

Koul, Anil, Arnoult, Eric, Lounis, Nacer, Guillemont, Jerome, Andries, Koen

Journal:

Year:

2011

Language:

english

File:

PDF, 1023 KB

english, 2011

17

New Anti-Tuberculosis Drugs in Clinical Development: An Overview

Guillemont, Jerome, Lieby-Muller, Frederic, Lounis, Nacer, Balemans, Wendy, Koul, Anil, Andries, Koen

Journal:

Current Bioactive Compounds

Year:

2009

Language:

english

File:

PDF, 374 KB

english, 2009

18

Synthesis and evaluation of analogues of the tuberculosis drug bedaquiline containing heterocyclic B-ring units

Choi, Peter J., Sutherland, Hamish S., Tong, Amy S.T., Blaser, Adrian, Franzblau, Scott G., Cooper, Christopher B., Lotlikar, Manisha U., Upton, Anna M., Guillemont, Jerome, Motte, Magali, Queguiner,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2017

Language:

english

File:

PDF, 896 KB

english, 2017

19

In Search of a Novel Anti-HIV Drug: Multidisciplinary Coordination in the Discovery of 4-[[4-[[4-[(1E)-2-Cyanoethenyl]-2,6-dimethylphenyl]amino]-2- pyrimidinyl]amino]benzonitrile (R278474, Rilpivirine)

Janssen, Paul A. J., Lewi, Paul J., Arnold, Eddy, Daeyaert, Frits, de Jonge, Marc, Heeres, Jan, Koymans, Luc, Vinkers, Maarten, Guillemont, Jérôme, Pasquier, Elisabeth

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 384 KB

english, 2005

20

A computational model of the inhibition of Mycobacterium tuberculosis ATPase by a new drug candidate R207910

Marc R. de Jonge, Luc H.M. Koymans, Jérôme E.G. Guillemont, Anil Koul, Koen Andries

Journal:

Proteins: Structure, Function, and Bioinformatics

Year:

2007

Language:

english

File:

PDF, 573 KB

english, 2007

21

Conformational Analysis of R207910, a New Drug Candidate for the Treatment of Tuberculosis, by a Combined NMR and Molecular Modeling Approach

Sandrine Gaurrand, Stéphanie Desjardins, Christophe Meyer, Pascal Bonnet, Jean-Michel Argoullon, Hassan Oulyadi, Jérôme Guillemont

Journal:

Chemical Biology & Drug Design

Year:

2006

Language:

english

File:

PDF, 229 KB

english, 2006

22

Crystal Structures for HIV-1 Reverse Transcriptase in Complexes with Three Pyridinone Derivatives: A New Class of Non-Nucleoside Inhibitors Effective against a Broad Range of Drug-Resistant Strains

Himmel, Daniel M., Das, Kalyan, Clark,, Arthur D., Hughes, Stephen H., Benjahad, Abdellah, Oumouch, Said, Guillemont, Jérôme, Coupa, Sophie, Poncelet, Alain, Csoka, Imre, Meyer, Christophe, Andries, K

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 636 KB

english, 2005

23

[1,2]-Wittig Rearrangement of (Benzyloxy)acetamides

Hameury, Thomas, Guillemont, Jérôme, Van Hijfte, Luc, Bellosta, Véronique, Cossy, Janine

Journal:

Year:

2008

Language:

english

File:

PDF, 86 KB

english, 2008

24

Ion mobility-mass spectrometry analysis of diarylquinoline diastereomers: Drugs used for tuberculosis treatment

Domalain, Virginie, Hubert-Roux, Marie, Quéguiner, Laurence, Fouque, Dany JD, Arnoult, Eric, Speybrouck, David, Guillemont, Jérôme, Afonso, Carlos

Journal:

European Journal of Mass Spectrometry

Year:

2018

Language:

english

File:

PDF, 960 KB

english, 2018

25

ChemInform Abstract: Diastereodivergent Addition of Allenylzincs to Aryl Glyoxylates.

Thomas Hameury, Jerome Guillemont, Luc Van Hijfte, Veronique Bellosta, Janine Cossy

Journal:

Year:

2009

File:

PDF, 33 KB

2009

26

A fit for purpose synthesis of (R)-2-methyl-azepane

Guizzetti, Sylvain, Michaut, Antoine, Federspiel, Guillaume, Eymard, Julien, Caron, Isabelle, Quatrevaux, Sabrina, Daras, Etienne, Jolly, Sandrine, Guillemont, Jerome, Lançois, David

Journal:

Organic Process Research & Development

Year:

2019

File:

PDF, 250 KB

2019

27

ChemInform Abstract: Reduction of Alkynyl α-Hydroxy Esters: Stereoselective α-Ketol Rearrangement.

Thomas Hameury, Veronique Bellosta, Jerome Guillemont, Luc Van Hijfte, Janine Cossy

Journal:

Year:

2010

File:

PDF, 44 KB

2010

28

3-Iodo-4-phenoxypyridinones (IOPY's), a new family of highly potent non-nucleoside inhibitors of HIV-1 reverse transcriptase

Abdellah Benjahad, Jérôme Guillemont, Koen Andries, Chi Hung Nguyen, David S Grierson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 155 KB

english, 2003

29

3-Iodo-4-phenoxypyridinones (IOPY′s), a New Family of Highly Potent Non-Nucleoside Inhibitors of HIV-1 Reverse Transcriptase.

Abdellah Benjahad, Jerome Guillemont, Koen Andries, Chi Hung Nguyen, David S. Grierson

Journal:

Year:

2004

File:

PDF, 87 KB

2004

30

Aldolisation-type reaction versus Michael-type addition. Hemiacetal vinylogs: Versatile synthons.

Pierre Duhamel, Jérôme Guillemont, Jean-Marie Poirier, Pierre Chabardes

Journal:

Tetrahedron Letters

Year:

1993

Language:

english

File:

PDF, 225 KB

english, 1993

31

Difluoromethylbenzoxazole Pyrimidine Thioether Derivatives: A Novel Class of Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors

Boyer, Jérémie, Arnoult, Eric, Médebielle, Maurice, Guillemont, Jérôme, Unge, Johan, Jochmans, Dirk

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 1.35 MB

english, 2011

32

ChemInform Abstract: Novel Procedure for the Coupling of Sterically Hindered Electron-Deficient Anilines to the 6-Position of the Purine Core.

Ruben Leenders, Jan Heeres, Dirk Vandenput, Jerome Guillemont, Paul Lewi

Journal:

Year:

2012

File:

PDF, 28 KB

2012

33

3-(Arylamino)-1,2,4-triazin-5-one: A Novel Synthesis and Its Use

Ruben Leenders, Jan Heeres, Dirk Vandenput, Remco Zijlmans, Jérôme Guillemont, Paul Lewi

Journal:

European Journal of Organic Chemistry

Year:

2010

Language:

english

File:

PDF, 92 KB

english, 2010

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